Kolexia
Azas Nadine
Pharmacien
Centre Hospitalier General La Ciotat
La Ciotat, France
80 Activités
2 Followers

Scientifique
Digital
Production scientifique
Activités par an
Expertise
Sujets de recherche
{{person.topmesh1.name}} Leishmaniose Paludisme Paludisme à Plasmodium falciparum Maladies parasitaires Toxoplasmose Maladie du sommeil Parasitémie Leishmaniose viscérale Infections à VIH

Industries

Sanofi
1 collaboration(s)
Dernière en 2017
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Dernières activités

Target fishing reveals PfPYK-1 and PfRab6 as potential targets of an antiplasmodial 4-anilino-2-trichloromethylquinazoline hit compound.
Bioorganic & medicinal chemistry   28 février 2024
Novel thienopyrimidones targeting hepatic and erythrocytic stages of Plasmodium parasites with increased microsomal stability.
European journal of medicinal chemistry   13 octobre 2023
New antiplasmodial 4-amino-thieno3,2-dpyrimidines with improved intestinal permeability and microsomal stability.
European journal of medicinal chemistry   13 janvier 2023
Design, Synthesis, and Antiprotozoal Evaluation of New Promising 2,9- (substituted-aminomethyl)-4,7-phenyl-1,10-phenanthroline Derivatives, a Potential Alternative Scaffold to Drug Efflux.
Pathogens (Basel, Switzerland)   13 novembre 2022
Improving Aqueous Solubility and In Vitro Pharmacokinetic Properties of the 3-Nitroimidazo1,2- pyridine Antileishmanial Pharmacophore.
Pharmaceuticals (Basel, Switzerland)   13 août 2022
Synthesis of antiplasmodial 2-aminothieno3,2-dpyrimidin-4(3H)-one analogues using the scaffold hopping strategy.
European journal of medicinal chemistry   20 juillet 2022
Pd-catalyzed C-C and C-N cross-coupling reactions in 2-aminothieno3,2- pyrimidin-4(3 )-one series for antiplasmodial pharmacomodulation.
RSC advances   08 juillet 2022
4-Substituted Thieno3,2- pyrimidines as Dual-Stage Antiplasmodial Derivatives.
Pharmaceuticals (Basel, Switzerland)   01 juillet 2022
Treating leishmaniasis in Amazonia, part 2: Multi-target evaluation of widely used plants to understand medicinal practices.
Journal of ethnopharmacology   05 février 2022
Challenges and Tools for In Vitro Exploratory Screening in the Drug Development Process: An Updated Review.
Pathogens (Basel, Switzerland)   10 décembre 2021